Translate

Search This Blog

Saturday, 13 September 2014

Paracetamol preparation

Chemical Structure  

Synonyms: Acetaminophen ; N-Acetyl-p-aminophenol ; N-(4-Hydroxyphenyl
 Theory

  Chemicals Required:
1.    para-Aminophenol : 6 g
2.     Acetic anhydride : 6.5 ml
3.    Concentrated Sulphuric acid : 4 drops.
Procedure:
1.    Weigh 6 g of para-aminophenol and transfer to a 100 ml thoroughly cleaned and dried conical flask.
2.    Add to the flask 6.5 ml of acetic anhydride and 3–4 drops of concentrated sulphuric acid cautiously.
3.    The contents of the flask may be mixed thoroughly. Warm the mixture on a waterbath previously maintained at 60°C for about 20–25 minutes with constant stirring.
4.    Allow the contents of the flask to attain room temperature, and pour it directly into a beaker having 100 ml of cold water (with a few chips of crushed ice) and stir it vigorously.
5.    The crude product obtained in (4) is filtered onto a Büchner funnel using suction,wash it with plenty of cold water, drain well and dry the product either between the folds of filter paper and air-dry it or dry it in an electric oven maintained at 100°C.
The yield of crude paracetamol (169–170.5°C) is approximately 6.8g.
 Recrystallisation: Dissolve the crude product in 70% (v/v) ethanol and warm it to 60°C ; add 2 g of powdered animal charcoal (decolourizing carbon). Filter and concentrate the filtrate over a water-bath. Allow it to cool and large crystals will separate out.
The yield of the pure paracetamol (mp 169–170.5°C) is 6.5 g.
 Uses
 antipyretic and analgesic.

No comments:

Post a Comment